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GENERAL
TITLE
CRYSTAL STRUCTURE OF TRIM24 PHD-BROMODOMAIN COMPLEXED WITH 2,4- DIMETHOXY-N-(1-METHYL-2-OXO-1,2,3,4-TETRAHYDROQUINOLIN-6-YL)BENZENE- 1-SULFONAMIDE (3B)
DATE LAST MODIFIED
9 Mar 2016
RELEASE
24 Jun 2015
OBSOLETE
CLASSIFICATION
TRANSCRIPTION/TRANSCRIPTION INHIBITOR
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
C 1 2 1
RESOLUTION RANGE HIGH
1.73
RESOLUTION RANGE LOW
60.73
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.5B00405
PDBe
Chains
Structure Chain | Target Protein | Gene | Expression System | Organism | Synonims | Actions |
---|---|---|---|---|---|---|
O15164 | TRIM24, RNF82, TIF1, TIF1A | ESCHERICHIA COLI | HUMAN | TIF1-ALPHA,E3 UBIQUITIN-PROTEIN LIGASE TRIM24,RING ... | Mutations | |
O15164 | TRIM24, RNF82, TIF1, TIF1A | ESCHERICHIA COLI | HUMAN | TIF1-ALPHA,E3 UBIQUITIN-PROTEIN LIGASE TRIM24,RING ... | Mutations |
NGL Viewer is used for the molecular visualization.
- AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
- AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402