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GENERAL
TITLE
CRYSTAL STRUCTURE OF THE TANDEM BROMODOMAIN (BD1, BD2) OF HUMAN TAF1 BOUND TO MTORC1/2 INHIBITOR AZD3147
DATE LAST MODIFIED
23 Mar 2022
RELEASE
22 Sept 2021
OBSOLETE
CLASSIFICATION
GENE REGULATION
EXPERIMENT TYPE
X-RAY DIFFRACTION
SPACE GROUP
P 21 21 21
RESOLUTION RANGE HIGH
2.2
RESOLUTION RANGE LOW
36.02
PUBMED ID
DOI
10.1021/ACS.JMEDCHEM.1C01999
LIGANDS

Chains

Structure ChainTarget ProteinGeneExpression SystemOrganismSynonimsActions
P21675 TAF1, BA2R, CCG1, CCGS, TAF2A ESCHERICHIA COLI HUMAN
CELL CYCLE GENE 1 PROTEIN,TBP-ASSOCIATED FACTOR 25 ...
Mutations
NGL Viewer is used for the molecular visualization.
  • AS Rose, AR Bradley, Y Valasatava, JM Duarte, A Prlić and PW Rose. NGL viewer: web-based molecular graphics for large complexes. Bioinformatics: bty419, 2018. doi:10.1093/bioinformatics/bty419
  • AS Rose and PW Hildebrand. NGL Viewer: a web application for molecular visualization. Nucl Acids Res (1 July 2015) 43 (W1): W576-W579 first published online April 29, 2015. doi:10.1093/nar/gkv402